Potentially Hepatotoxic Drugs

Potentially Hepatotoxic Drugs

Finding

Drug

Hepatocellular: Elevated ALT

AcarboseAcarbose

AcetaminophenAcetaminophen

AllopurinolAllopurinol

AmiodaroneAmiodarone

Antiretroviral therapy drugs

BupropionBupropion

FluoxetineFluoxetine

Germander

Green tea extractGreen tea extract

BaclofenBaclofen

IsoniazidIsoniazid

Kava

KetoconazoleKetoconazole

LisinoprilLisinopril

LosartanLosartan

MethotrexateMethotrexate

NSAIDs

OmeprazoleOmeprazole

PD-1/PD-L1 inhibitors

ParoxetineParoxetine

PyrazinamidePyrazinamide

RifampinRifampin

RisperidoneRisperidone

SertralineSertraline

Statins

Tetracyclines

TrazodoneTrazodone

Trovafloxacin

Valproate

Cholestatic: Elevated alkaline phosphatase and total bilirubin

Amoxicillin/clavulanateAmoxicillin/clavulanate

Anabolic steroids

ChlorpromazineChlorpromazine

ClopidogrelClopidogrel

Oral contraceptives

Erythromycins

Estrogens

IrbesartanIrbesartan

MirtazapineMirtazapine

Phenothiazines

TerbinafineTerbinafine

Tricyclic antidepressants

Mixed: Elevated alkaline phosphatase and ALT

AmitriptylineAmitriptyline

AzathioprineAzathioprine

CaptoprilCaptopril

CarbamazepineCarbamazepine

ClindamycinClindamycin

CyproheptadineCyproheptadine

EnalaprilEnalapril

NitrofurantoinNitrofurantoin

PhenobarbitalPhenobarbital

PhenytoinPhenytoin

Sulfonamides

TrazodoneTrazodone

Trimethoprim/sulfamethoxazoleTrimethoprim/sulfamethoxazole

VerapamilVerapamil

ALT = alanine aminotransferase; AST= aspartate aminotransferase; NSAID = nonsteroidal anti-inflammatory drug.

ALT = alanine aminotransferase; AST= aspartate aminotransferase; NSAID = nonsteroidal anti-inflammatory drug.